Peptide Active Data Details
Basic Peptide Information
DICL ID
DICL_Pep_03985
Ion Channel
Neuronal acetylcholine receptor subunit alpha-7
Peptide Function
Blocker
Gene Name
CHRNA7
Activity Data (nM)
IC50
0.539 nM
Ki
Not available
EC50
Not available
Kd
Not available
Biologically Active
Not specified
Sequence Information
Peptide Sequence
DECCSNPACRLNNPHVCRRR
Peptide UniProt Accession
Not available
UniParc
UPI000DC0C663
Peptide Synonyms/Alias
ArIB[V11L]
Peptide Species
Not specified
Peptide Name
Not available
CAS Number
Not available
Experimental Conditions
pH
pH 7.1 to 7.5
Holding Potential (mV)
−70 mV
Temperature
~22 °C
Test Method
Patch-clamping
Test Species
Xenopus laevis oocyte
Binding Information
Binding Site
Not specified
Binding Site Residue
Not specified
Ion Channel Information
Gene Abbreviation (ABB)
nAChRs
Ion Channel UniProt Accession
Source Organism
Homo sapiens (Human)
References & Disease Information
Disease
Not specified
PubChem CID
Not available
URL
Not available
PMID
Patent
Not available